1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. Src
  4. Src Inhibitors

Src Inhibitors

Lck

Fyn

Blk

Fgr

Hck

Lyn

Yes

SRC-3

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Src Degraders & Inhibitors
Product Name Lck Fyn Blk Fgr Hck Lyn Yes SRC-3 Purity
PRT062607 Hydrochloride
Lck, IC50: 249 nM ([2])
              98.07%
GLPG3312
Lck, IC50: 385 nM
Fyn, IC50: 447 nM
Blk, IC50: 730 nM
 
Hck, IC50: 2511 nM
Lyn, IC50: 272 nM
Yes, IC50: 598 nM
  98.57%
Velzatinib
Lck, IC50: 141 nM
              99.40%
AZM475271
Lck, IC50: 0.03 μM
              99.89%
SB 220025
p56-Lck, IC50: 3.5 μM
              99.90%
PRT062607 acetate
Lck, IC50: 249 nM ([2])
              99.83%
RK-20448
Lck, IC50: 0.24 μM
Fyn, IC50: 2.03 μM
Blk, IC50: 0.37 μM
          99.38%
Lck-IN-2
Lck, IC50: 10.6 nM
             
SJ11646
Lck, DC50: 0.00838 pM
             
Antifibrotic agent 1
Lck
Fyn
   
Hck
Lyn
Yes
 
MRT-10350        
Hck
     
MRT-7612
Lck
     
Hck
Lyn
   
BY13              
SRC-3, DC50: 0.031 μM
N-Deshydroxyethyl Dasatinib-C3-NH2
Lck
             
LCK degrader-2
Lck
             
SIK1-IN-1
Lck, IC50: 3.7 nM
   
Fgr, IC50: <3 nM
Hck, IC50: <3 nM
Lyn, IC50: <1.5 nM
Yes, IC50: <3 nM
 
BMS-243117
Lck, IC50: 4 nM
Fyn, IC50: 32 nM
Blk, IC50: 84 nM