2. GPCR/G Protein
  3. GHSR
  4. CP-464709

CP-464709 是一种可穿透血脑屏障的 Ghrelin 受体激动剂。CP-464709 通过激活脊髓交感节前神经元引起血压升高。CP-464709 静脉给药引起双相血压反应，鞘内给药仅引起升压。CP-464709 可用于心血管疾病的研究。

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CP-464709

CP-464709 Chemical Structure

CAS No. : 193272-70-7

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CP-464709 相关抗体

Top Publications Citing Use of Products

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GHSR1a

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CP-464709 is a Ghrelin receptor agonist that can penetrate the blood-brain barrier. CP-464709 causes an increase in blood pressure by activating pre sympathetic neurons in the spinal cord. CP-464709 causes biphasic blood pressure response when administered intravenously, while intrathecal administration only causes pressor. CP-464709 can be used for research on cardiovascular conditions[1].

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
Pituitary gland cell EC50
3 nM
Compound: 4, (CP-464709-18)
In vitro effective concentration required for 50% stimulation of GH release in rat pituitary cell cultures.
In vitro effective concentration required for 50% stimulation of GH release in rat pituitary cell cultures.
[PMID: 12392732]
分子量

610.58

Formula

C28H31F5N6O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CP-464709 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CP-464709193272-70-7CP464709CP 464709GHSRGrowth hormone secretagogue receptorGhrelin receptorGhrelinblood pressurecardiovascularInhibitorinhibitorinhibit

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产品名称：
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目录号：
HY-19454
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