2. Metabolic Enzyme/Protease
  3. Cytochrome P450
  4. CYP3A4-IN-6

CYP3A4-IN-6 (Compound 8a) 是一种具有组织选择性代谢的 CYP3A4 抑制剂。CYP3A4-IN-6 在肠道 S9 组分存在下保持稳定，而在肝脏 S9组分中迅速代谢，形成活性较低的代谢物。CYP3A4-IN-6 可用于肠道选择性研究。

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CYP3A4-IN-6

CYP3A4-IN-6 Chemical Structure

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CYP3A4-IN-6 相关抗体

Top Publications Citing Use of Products

查看 Cytochrome P450 亚型特异性产品:

查看所有亚型
CYP1 CYP2 CYP3 CYP4 CYP11 CYP17 Aromatase/CYP19A1 CYP26 CYP51 CYP1A2 CYP2D6 CYP2C9 CYP2C19 CYP3A4 CYP17A1

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CYP3A4-IN-6 (Compound 8a) is a CYP3A4 inhibitor with tissue-selective metabolism. CYP3A4-IN-6 remains stable in the intestinal S9 component but is rapidly metabolized in the liver S9 component, forming a less active metabolite. CYP3A4-IN-6 can be used for intestinal selectivity studies[1].

IC50 & Target[1]

CYP3A4

 

分子量

322.36

Formula

C19H18N2O3
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CYP3A4-IN-6 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CYP3A4-IN-6Cytochrome P450CYPsAntedrugCytochrome P450 inhibitorPharmacokinetic boosterImidazoleStructure-activity relationshipInhibitorinhibitorinhibit

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产品名称：
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目录号：
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