2. Anti-infection Metabolic Enzyme/Protease
  3. Antibiotic Carbonic Anhydrase Bacterial
  4. Dealanylascamycin

Dealanylascamycin (AT-265) (Compound 2) 是一种核苷类抗生素。AT 265 是碳酸酐酶 (CA) 抑制剂，对 hCA I、hCA II、hCA IV 和 hCA IX 的 Ki 值分别为 167、65.2、234 和 143 nM。Dealanylascamycin 是 Ascamycin (HY-121071) 的活性形式。Dealanylascamycin 具有广谱抗菌性，对 Xanthomonas citri (MIC = 0.4 μg/mL) 等病原菌均有效。Dealanylascamycin 具有高细胞毒性。

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Dealanylascamycin

Dealanylascamycin Chemical Structure

CAS No. : 66522-52-9

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Dealanylascamycin 相关抗体

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Aminoglycoside Glycopeptide Lipopeptide Macrolide Oxazolidinone Quinolone Tetracycline β-lactam

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  • 生物活性

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  • 参考文献

生物活性

Dealanylascamycin (AT-265) (Compound 2) is a nucleoside antibiotic. AT 265 is a carbonic anhydrase (CA) inhibitor, with Ki values of 167, 65.2, 234, and 143 nM for hCA I, hCA II, hCA IV, and hCA IX respectively. Dealanylascamycin is the active form of Ascamycin (HY-121071). Dealanylascamycin exhibits broad-spectrum antibacterial activity and is effective against pathogenic bacteria such as Xanthomonas citri (MIC = 0.4 μg/mL). Dealanylascamycin has high cytotoxicity[1][2].

IC50 & Target[1]

hCA I

167 nM (Ki)

hCA II

65.2 nM (Ki)

hCA IX

143 nM (Ki)

分子量

380.76

Formula

C10H13ClN6O6S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Dealanylascamycin 相关分类

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Keywords:

Dealanylascamycin66522-52-9AT-265AT265AT 265AntibioticCarbonic AnhydraseBacterialCarbonate dehydrataseNucleoside antibioticSulfamoyl chloride adenosineCarbonic anhydrase inhibitionX-ray crystallographyAntimicrobial activityStructure-activity relationshipSelective toxicityInhibitorinhibitorinhibit

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