2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. Fadolmidine hydrochloride

Fadolmidine hydrochloride 是一种新型选择性 α2 肾上腺素受体 (α2-AR) 激动剂，对 2A、2B 和 2C 亚型的 EC50 值分别为 0.4 nM、4.9 nM 和 0.5 nM。Fadolmidine hydrochloride 对多种疼痛类型有效，例如热痛、机械痛和内脏痛。此外，Fadolmidine hydrochloride 还能抑制大鼠输精管的电刺激诱导收缩。

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Fadolmidine hydrochloride

Fadolmidine hydrochloride Chemical Structure

CAS No. : 189353-32-0

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Other Forms of Fadolmidine hydrochloride:

Fadolmidine hydrochloride 相关抗体

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生物活性

Fadolmidine hydrochloride is a novel, selective α2-adrenoceptor (α2-AR) agonist with EC50 values of 0.4 nM, 4.9 nM and 0.5 nM for 2A, 2B and 2C, respectively. Fadolmidine hydrochloride has been effective against various submodalities of pain such as heat pain, mechanical pain, and visceral pain. Fadolmidine hydrochloride inhibits also electrically evoked contractions in rat vas deferens[1][2].

IC50 & Target[1]

α2-adrenergic receptor

 

分子量

250.72

Formula

C13H15ClN2O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Fadolmidine hydrochloride 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Fadolmidine189353-32-0Adrenergic ReceptorBeta Receptorheat painmechanical painand visceral painInhibitorinhibitorinhibit

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产品名称：
Fadolmidine hydrochloride
目录号：
HY-106388A
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