2. GPCR/G Protein
  3. P2Y Receptor
  4. MRS4654

MRS4654 是一种高效、中性的 P2Y14R (hP2Y14R IC50 = 15.0 nM，mP2Y14R IC50 = 18.6 nM) 拮抗剂。MRS4654 具有镇痛和抗炎效果。MRS4654 可以用于哮喘和神经性疼痛的研究。

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MRS4654

MRS4654 Chemical Structure

CAS No. : 2765570-58-7

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MRS4654 相关抗体

Top Publications Citing Use of Products

查看 P2Y Receptor 亚型特异性产品:

查看所有亚型
P2Y1 Receptor P2Y2 Receptor P2Y6 Receptor P2Y12 Receptor P2Y13 Receptor P2Y14 Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

MRS4654 is an efficient and neutral P2Y14R (hP2Y14R IC50 = 15.0 nM, mP2Y14R IC50 = 18.6 nM) antagonist. MRS4654 has analgesic and anti-inflammatory effects. MRS4654 can be used for research on asthma and neuropathic pain[1].

IC50 & Target[1]

hP2Y14R

15 nM (IC50)

mP2Y14R

18.6 nM (IC50)

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
HepG2 IC50
8.47 μM
Compound: 32
Cytotoxicity against human HepG2 cells
Cytotoxicity against human HepG2 cells
[PMID: 33787273]
分子量

489.44

Formula

C28H18F3NO4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

MRS4654 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MRS46542765570-58-7MRS 4654MRS-4654P2Y ReceptorP2Y14Ranalgesicanti-inflammatoryasthmaneuropathic painInhibitorinhibitorinhibit

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产品名称：
MRS4654
目录号：
HY-156220
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