2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor Adrenergic Receptor
  4. Pelanserin

Pelanserin (Compound 1) 是一种口服有效的降压剂。Pelanserin 是一种强效的 5-HT2 受体 (5-HT2 receptor) 拮抗剂。Pelanserin 具有阻断 α-肾上腺素能受体 (α-adrenergic receptor) 活性，其 ED50 为 0.03 μg/mL。Pelanserin 具有血管舒张活性，其 ED100 为 5 μg。Pelanserin 在高血压大鼠和肾性高血压犬种均具有抗高血压活性。Pelanserin 可用于研究高血压。

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Pelanserin

Pelanserin Chemical Structure

CAS No. : 2208-51-7

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Pelanserin 相关抗体

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5-HT Receptor 5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Pelanserin (Compound 1) is an orally active antihypertensive agent. Pelanserin is a potent 5-HT2 receptor antagonist. Pelanserin has the ability to block the activity of α-adrenergic receptor, with its ED50 being 0.03 μg/mL. Pelanserin has vasodilatory activity, with its ED100 being 5 μg. Pelanserin exhibits antihypertensive activity in hypertensive rats and renal hypertensive dog breeds. Pelanserin can be used for research on hypertension[1][2][3].

分子量

364.44

Formula

C21H24N4O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Pelanserin 相关分类

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Pelanserin2208-51-75-HT ReceptorAdrenergic ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorBeta ReceptorQuinazolinedionesvasodilatorsantihypertensive agentsalpha-adrenergic blockadestructure-activity relationshipInhibitorinhibitorinhibit

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