2. GPCR/G Protein
  3. Taste Receptor
  4. S7958

S7958 是一种选择性的和口服有效的 TAS2R8 苦味受体拮抗剂，其 IC50 为 0.06 μM。S7958 仅对 TASR8 和 TAS2R39 有微弱抑制，对其他受体无显著影响。S7958 通过选择性拮抗人体苦味受体 TAS2R8，显著抑制由咖啡、药物活性成分 (API) 等物质引起的苦味感知。S7958 可在医疗领域用于改善口服制剂的苦味研究。

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S7958

S7958 Chemical Structure

CAS No. : 1217341-48-4

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S7958 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

S7958 is a selective and orally active antagonist of the TAS2R8 bitter taste receptor, with its IC50 being 0.06 μM. S7958 only has a weak inhibitory effect on TASR8 and TAS2R39, and has no significant impact on other receptors. S7958 significantly inhibits the perception of bitterness caused by substances such as coffee and drug active ingredients (API) by selectively antagonizing the human bitter taste receptor TAS2R8. S7958 can be used in the medical field to improve the research on the bitterness of oral preparations[1].

分子量

409.44

Formula

C21H23N5O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

S7958 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

S79581217341-48-4S 7958S-7958Taste Receptorbitterness maskingstructure-activity relationshiphydantoin derivativessensory evaluationInhibitorinhibitorinhibit

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产品名称：
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目录号：
HY-139898
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