Preparation and suzuki-miyaura coupling reactions of tetrahydropyridine-2-boronic acid pinacol esters

EG Occhiato, F Lo Galbo, A Guarna

文献索引：Occhiato, Ernesto G.; Lo Galbo, Fabrizio; Guarna, Antonio Journal of Organic Chemistry, 2005 , vol. 70, # 18 p. 7324 - 7330

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被引用次数: 50

摘要

A study on the conversion of lactam-derived vinyl triflates and phosphates into the corresponding vinyl boronates was carried out. While δ-valerolactam-derived vinyl triflates were successfully converted into 1, 4, 5, 6-tetrahydropyridine-2-boronic acid pinacol ester ...

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