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1428630-86-7生产厂家
1428630-86-7价格
化源商城直购
rat mGluR5:9.3 nM (EC50)
rat mGluR5:8.03 nM (pEC50)
[1]. Turlington M, Noetzel MJ, Chun A, et al. Exploration of allosteric agonism structure-activity relationships within an acetylene series of metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulators (PAMs): discovery of 5-((3-fluorophenyl)ethynyl)-N-(3-methyloxetan-3-yl)picolinamide (ML254). J Med Chem. 2013;56(20):7976-7996.