产品货号:A101210
产品名称:A 83-01
Synonyms:3-(6-Methyl-2-pyridinyl)-N-phenyl-4-(4-quinolinyl)-1H-pyrazole-1-carbothioamide
CAS号:909910-43-6
分子式:C₂₅H₁₉N₅S
Appearance:Off-White to Pale Yellow Solid
Melting Point:207-209°C
分子量:421.52
Storage:4°C, Hygroscopic
Solubility:Chloroform (Slightly), DMSO (Slightly), Methanol (Very Slightly)
Stability
Hygroscopic, Moisture Sensitive
Category:Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
应用:A 83-01 is a selective inhibitor of TGF-b type I receptor. A 83-01 treatment increases tumor permeability.
参考文献:Minowa, T. et al.: British. J. Canc., 101, 1884 (2009)
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