2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor Dopamine Receptor
  4. Setoperone

Setoperone 是一种口服有效的、强效的 5-HT₂ 受体 (5-HT₂ receptor) 拮抗剂和中度的多巴胺 D₂ 受体 (D₂ receptor) 阻断剂。Setoperone 从受体解离的速度较快，但其在体内容易被血清素受体“捕获”，导致洗脱后仍存在持续性受体抑制。Setoperone 可用于研究 II 型精神分裂症的阴性症状及伴发情绪障碍。

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Setoperone

Setoperone Chemical Structure

CAS No. : 86487-64-1

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Setoperone 相关抗体

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查看 5-HT Receptor 亚型特异性产品:

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5-HT Receptor 5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Setoperone is an orally active and potent 5-HT₂ receptor antagonist and a moderate dopamine D₂ receptor blocker. Setoperone dissociates from the receptors relatively quickly, but it is easily "captured" by serotonin receptors in the body, resulting in persistent receptor inhibition even after elution. Setoperone can be used to study the negative symptoms of type II schizophrenia and associated mood disorders[1][2].

分子量

401.50

Formula

C21H24FN3O2S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Setoperone 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Setoperone86487-64-15-HT ReceptorDopamine ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorSerotonin antagonismDopamine blockadeSchizophrenia5-HT? receptorsD? receptorsBPRSExtrapyramidal symptomsReceptor down-regulationChronic treatmentInhibitorinhibitorinhibit

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