Chemsrc provides Others's classification, including all related biologically active compounds cover the research fields of cancer, neuroscience, immunology and other popular diseases, etc.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Biotin NHS

Biotin NHS is an amino reactive biotin reagent used in the preparation of biotinylated surfaces or polypeptides.

  • CAS Number: 35013-72-0
  • MF: C14H19N3O5S
  • MW: 341.383
  • Catalog: Dye Reagents
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: 212-214 °C
  • Flash Point: N/A

Boc-Gly-Lys-Arg-AMC

Boc-Gly-Lys-Arg-AMC is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development[1].

  • CAS Number: 109358-48-7
  • MF: C29H44N8O7
  • MW: 616.71
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(+)-Scandine

Scandine is a alkaloid compound isolated from the twigs and leaves of Melodinus suaveolens[1].

  • CAS Number: 24314-59-8
  • MF: C21H22N2O3
  • MW: 350.411
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 521.4±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 269.1±30.1 °C

4-oxo-4-HPR

4-Oxofenretinide (4-Oxo-4-HPR) is a metabolite of Fenretinide (HY-15373). 4-Oxofenretinide induces cell growth inhibition in ovarian, breast, and neuroblastoma tumor cell lines. 4-Oxofenretinide causes a marked accumulation of cells in G2-M. 4-Oxofenretinide induces cancer cell apoptosis through caspase-9[1].

  • CAS Number: 865536-65-8
  • MF: C26H31NO3
  • MW: 405.53
  • Catalog: Apoptosis
  • Density: 1.131g/cm3
  • Boiling Point: 641.8ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 341.9ºC

β-Tomatine

β-Tomatine is a breakdown product of a-tomatine and a less fungitoxic compound. β-Tomatine can suppress plant defense responses[1].

  • CAS Number: 17406-46-1
  • MF: C45H75NO17
  • MW: 902.07300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Encecalin

Encecalin is a natural benzofuran compound[1].

  • CAS Number: 20628-09-5
  • MF: C14H16O3
  • MW: 232.275
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 367.7±42.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 167.6±14.3 °C

DSPE-PEG-Mal

DSPE-PEG-Maleimide has DSPE phospholipid and maleimide to prepare nanostructured lipid carrier. DSPE-PEG-Maleimide extends blood circulation time and higher stability for encapsulated drugs[1][2].

  • CAS Number: 474922-22-0
  • MF: C139H271N4O67P
  • MW: 2941.61
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

TNIK-IN-7

TNIK-IN-7 (Compound 8) is an inhibitor of Traf2 and Nck-interacting kinase (TNIK), with IC50 of 11 nM, that has antitumor activity[1].

  • CAS Number: 1417795-24-4
  • MF: C23H22N4O2
  • MW: 386.4
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

D-Tetramannuronic acid

D-Tetramannuronic acid, an alginate oligomer, is produced by marine brown algae and by a limited range of Gram negative bacteria. D-Tetramannuronic acid can be used for the research of pain and vascular dementia[1][2][3][4].

  • CAS Number: 149511-34-2
  • MF: C24H34O25
  • MW: 722.51
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

METHYL 2-(CYCLOPENTYLAMINO)ACETATE HYDROCHLORIDE

Methyl 2-(cyclopentylamino)acetate hydrochloride is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 195877-46-4
  • MF: C8H16ClNO2
  • MW: 193.671
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Ontorpacept

Ontorpacept (TTI-621) is a soluble fusion protein that consists of the human SIRPα N-terminal (1-118) linked to the Fc region of human IgG1. The N-terminal (1-118)-fragment of ontorpacept is a binding domain for CD47 which is an inhibitor of phagocytosis by macrophages. Ontorpacept is a CD47-blocking checkpoint inhibitor with antitumor activity[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

w-Conotoxin SVIB

w-Conotoxin SVIB is a peptide toxin, it can be isolated from Conus venoms. w-Conotoxin SVIB inhibits twitch response with an IC50 value of 37 nM. w-Conotoxin SVIB induces respiratory distress and it can be lethal to mice at a high concentration[1][2].

  • CAS Number: 150433-82-2
  • MF: C105H176N38O36S6
  • MW:
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(-)-Gallocatechin

(-)-Gallocatechin, an epimer of (-)-Epigallocatechin (EGC), is contained in various tea products. (-)-Gallocatechin has antioxidant activities[1][2][3].

  • CAS Number: 3371-27-5
  • MF: C15H14O7
  • MW: 306.267
  • Catalog: Metabolic Disease
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 685.6±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 368.5±31.5 °C

propranolol

Propranolol is a noncardioselective β-blocker. Propranolol has membrane-stabilizing properties, but does not own intrinsic sympathomimetic activity. Propranolol hydrochloride is used to control hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy[1].

  • CAS Number: 525-66-6
  • MF: C16H21NO2
  • MW: 259.34300
  • Catalog: Cardiovascular Disease
  • Density: 1.093 g/cm3
  • Boiling Point: 434.9ºC at 760 mmHg
  • Melting Point: 163-164ºC
  • Flash Point: 216.8ºC

1,3,6-Trihydroxy-2-methylanthraquinone 3-O-alpha-L-rhamnosyl-(1->2)-beta-D-glucoside

2-Methyl-1,3,6-trihydroxy-9,10-anthraquinone 3-O-α-rhamnosyl-(1→2)-β-glucoside is anthraquinone glycoside found in the dried roots of Rubia cordifolia[1].

  • CAS Number: 87686-88-2
  • MF: C27H30O14
  • MW: 578.519
  • Catalog: Others
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 911.5±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 303.8±27.8 °C

Briquilimab

Briquilimab (JSP-191) is a non-toxic humanized monoclonal antibody targeting CD117 (c-Kit) to deplete hematopoietic stem cell (HSC). Briquilimab has safety to clear host marrow niche space to enable sufficient donor HSC engraftment and immune reconstitution as primary method of severe combined immunodeficiency (SCID)[1].

  • CAS Number: 2574591-89-0
  • MF:
  • MW:
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Undecylprodigiosin

Undecylprodigiosin is a cytotoxic immunosuppressant[1].

  • CAS Number: 52340-48-4
  • MF: C25H35N3O
  • MW: 393.56500
  • Catalog: Inflammation/Immunology
  • Density: 1.06g/cm3
  • Boiling Point: 589.8ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: N/A

EA-230

EA-230 is a synthetic oligopeptide originally derived from beta-human chorionic gonadotropin (beta-hCG) lysates. EA-230 has anti-inflammatory effects and can be used for the research of sepsis[1].

  • CAS Number: 503844-09-5
  • MF: C15H27N5O6
  • MW: 373.40500
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Benzyl(2R)-3-N,N-dibenzylamino-2-fluoropropanoate-13C3

Benzyl(2R)-3-N,N-dibenzylamino-2-fluoropropanoate-13C3 is a 13C-labeled and deuterium labeled Benzyl(2R)-3-N,N-dibenzylamino-2-fluoropropanoate[1].

  • CAS Number: 1217853-98-9
  • MF: C2113C3H24FNO2
  • MW: 380.43
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Tafluprost ethyl amide

Tafluprost ethyl amide is a prostaglandin derivative. Tafluprost ethyl amide is capable of intraocular pressure (IOP) reduction and influencing eyelash growth. Tafluprost ethyl amide can be used in antiglaucoma ophthalmic compositions or cosmetics[1].

  • CAS Number: 1185851-52-8
  • MF: C24H33F2NO4
  • MW: 437.520
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 609.3±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 322.3±31.5 °C

Fmoc-Asn-OH

Fmoc-Asn-OH is an asparagine derivative[1].

  • CAS Number: 71989-16-7
  • MF: C19H18N2O5
  • MW: 354.357
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 678.6±55.0 °C at 760 mmHg
  • Melting Point: 190 °C (dec.)(lit.)
  • Flash Point: 364.2±31.5 °C

Bisdemethoxycurcumin

Bisdemethoxycucurmin (p,p'-Dihydroxydicinnamoylmethane), a curcuminoid, has antioxidant and antiinflammatory activities[1][2].

  • CAS Number: 24939-16-0
  • MF: C19H16O4
  • MW: 308.328
  • Catalog: Inflammation/Immunology
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 551.3±45.0 °C at 760 mmHg
  • Melting Point: 91-93℃
  • Flash Point: 301.3±25.2 °C

WM382

WM382 is an orally active and potent dual plasmepsin IX/X (PMIX/X) inhibitor with IC50 values of 1.4 nM and 0.03 nM, respectively. WM382 has robust in vivo efficacy at multiple stages of the malaria parasite life cycle and an excellent resistance profile[1][2][3].

  • CAS Number: 2606990-92-3
  • MF: C29H36N4O4
  • MW: 504.62
  • Catalog: Infection
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

IBS008738

IBS008738 is a potent TAZ activator. IBS008738 stabilizes TAZ, increases the unphosphorylated TAZ level, enhances the association of MyoD with the myogenin promoter, upregulates MyoD-dependent gene transcription, and competes with myostatin in C2C12 cells. IBS008738 enhances myogenesis in C2C12 cells and facilitates muscle repair in a muscle injury model[1][2].

  • CAS Number: 385425-03-6
  • MF: C22H22N4O2
  • MW: 374.44
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

dl-4-hydroxyphenylglycine

2-Amino-2-(4-hydroxyphenyl)acetic acid is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 938-97-6
  • MF: C8H9NO3
  • MW: 167.16200
  • Catalog: Others
  • Density: 1.411g/cm3
  • Boiling Point: 446.3ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 223.7ºC

Ara-G

9-β-D-Arabinofuranosylguanine is a Guanosine (HY-N0097) analog and shows high affinity for deoxyguanosine kinase (dGK) with a Km of 8.0 μM. 9-β-D-Arabinofuranosylguanine can be used for the research of T-cell lymphoblastic disease[1][2].

  • CAS Number: 38819-10-2
  • MF: C10H13N5O5
  • MW: 283.241
  • Catalog: Cancer
  • Density: 2.3±0.1 g/cm3
  • Boiling Point: 775.9ºC at 760 mmHg
  • Melting Point: 225°C(lit.)
  • Flash Point: 423.1ºC

H-D-Phe(4-F)-OH.HCl

H-D-Phe(4-F)-OH.HCl is a phenylalanine derivative[1].

  • CAS Number: 122839-52-5
  • MF: C9H11ClFNO2
  • MW: 219.641
  • Catalog: Others
  • Density: 1.293g/cm3
  • Boiling Point: 313.3ºC at 760mmHg
  • Melting Point: 245 °C (dec.)(lit.)
  • Flash Point: 143.3ºC

Fmoc-D-Dbu(N3)-OH

Fmoc-D-Dbu(N3)-OH is a click chemistry reagent containing an Azide[1].

  • CAS Number: 1932023-47-6
  • MF: C19H18N4O4
  • MW: 366.37
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Head activator

Head activator neuropeptide is a mitogen for mammalian cell lines of neuronal or neuroendocrine origin. Head activator neuropeptide signals by binding GPR37 and stimulates cells to enter mitosis[1].

  • CAS Number: 79943-68-3
  • MF: C54H84N12O14
  • MW: 1125.32000
  • Catalog: Cancer
  • Density: 1.271g/cm3
  • Boiling Point: 1506.5ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 864.9ºC

Favezelimab

Favezelimab (MK-4280) is a humanized anti-LAG-3 monoclonal antibody that blocks the interaction between LAG-3 and its ligand MHC class II. Favezelimab has the potential for colorectal cancer (CRC) research combined with the PD-L1 inhibitor Pembrolizumab (HY-P9902)[1][2].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A