CAS号英文名称中文名称分子式分子量
228559-41-9KI 8751Ki8751 C24H18F3N3O4469.41263628006
623142-96-1Ki20227N-[4-[(6,7-二甲氧基-4-喹啉基)氧基]-2-甲氧基苯基]-N'-[1-(2-噻唑基)乙基]脲C24H24N4O5S480.536164283752
1100598-32-0Tepotinib特泊替尼C29H28N6O2492.571625709534
529-59-9Genistin染料木苷C21H20O10432.377507209778
697235-39-5EpisilvestrolEpisilvestrol C34H38O13654.657731533051
417716-92-8Lenvatinib乐伐替尼C21H19ClN4O4426.8530
796967-16-3LinifanibN-[4-(3-氨基-1H-吲唑-4-基)苯基]-N'-(2-氟-5-甲基苯基)脲C21H18FN5O375.398927211761
65678-07-1AG1024AG1024 抑制剂C14H13BrN2O305.169822454453
1202757-89-8SpebrutinibAVL-292C22H22FN5O3423.440187931061
897383-62-9AST-1306N-[4-[[3-氯-4-[(3-氟苯基)甲氧基]苯基]氨基]-6-喹唑啉基]-2-丙烯酰胺C24H18ClFN4O2448.876727581024
873305-35-2AIM-1005,6-二苯基-N-[[(2S)-四氢-2-呋喃基]甲基]呋喃并[2,3-D]嘧啶-4-胺C23H21N3O2371.431745290756
1002304-34-8AMG-2087-甲氧基-4-[(6-苯基-1,2,4-三唑并[4,3-B]哒嗪-3-基)甲氧基]喹啉C22H17N5O2383.402683973312
153436-53-4AG-1478次黄嘌呤.6-羟基嘌呤C16H14ClN3O2315.754262447357
1197958-12-5Alk-IN-15-氯-N2-[4-[4-(二甲基氨基)-1-哌啶基]-2-甲氧基苯基]-N4-[2-(二甲基亚膦酰)苯基]-2,4-嘧啶二胺C26H34ClN6O2P529.013925075531
811803-05-1Apatinib阿帕替尼C24H23N5O.CH4O3S493.57798
913376-83-7AMG-458盐酸米托蒽醌C30H29N5O5539.581766843796
319460-85-0Axitinib阿西替尼C22H18N4OS386.469522953033
439081-18-2BIBW 2992阿法替尼C24H25ClFN5O3485.938407659531
1050500-29-2Allitinib tosylate艾力替尼C31H26ClFN4O5S621.078348636627
1097917-15-1ASP3026N2-[2-甲氧基-4-[4-(4-甲基-1-哌嗪基)-1-哌啶基]苯基]-N4-[2-[(1-甲基乙基)磺酰基]苯基]-1,3,5-三嗪-2,4-二胺C29H40N8O3S580.744704246521
497839-62-0AEE788AEE788 (NVP-AEE788) 抑制剂C27H32N6440.583185195923
937265-83-3ARRY-380 analog6-[5-[[[2-(甲磺酰基)乙基]氨基]甲基]-2-呋喃基]-N-[3-甲基-4-([1,2,4]三唑并[1,5-A]吡啶-7-氧基)苯基]-4-氨基喹唑C29H27N7O4S569.634184122086
453562-69-1Motesanib莫特塞尼C22H23N5O373.450924158096
790299-79-5Masitinib马赛替尼C28H30N6OS498.642404079437
850879-09-3AmuvatinibN-(1,3-苯并二氧戊环-5-基甲基)-4-苯并呋喃并[3,2-d]嘧啶-4-基-1-哌嗪硫代甲酰胺C23H21N5O3S447.509543180466
875337-44-3MGCD-265 analog氟培龙C26H20FN5O2S2517.597705841064
1001917-37-8MK-80333-(1-甲基-1H-吡唑-4-基)-5-氧代-N-(2-吡啶甲基)-5H-苯并[4,5]环己烯并[1,2-B]吡啶-7-甲磺酰胺C25H21N5O3S471.530943632126
857876-30-3Motesanib diphosphate二磷酸莫替沙尼C22H29N5O9P2569.441286802292
366017-09-6Mubritinib木利替尼C25H23F3N4O2468.470936059952
917879-39-1MK-2461C24H25N5O5S495.550803899765
1092499-93-8NVP-BSK805NVP-BSK805 抑制剂C27H28F2N6O490.547632217407
940310-85-0NVP-BHG7124-甲基-3-[[1-甲基-6-(3-吡啶基)-1H-吡唑并[3,4-d]嘧啶-4-基]氨基]-N-[3-(三氟甲基)苯基]苯甲酰胺C26H20F3N7O503.478514671326
475489-16-8NVP-AEW541AVP-AEW541 抑制剂C27H29N5O439.552065610886
698387-09-6Neratinib来那替尼C30H29ClN6O3557.042665243149
1185763-69-2NVP-BVU972NVP-BVU972 抑制剂C20H16N6340.381242752075
475488-23-4NVP-ADW7425-(3-苄氧基苯基)-7-[反式-3-[(吡咯烷-1-基)甲基]环丁基]-7H-吡咯并[2,3-d]嘧啶-4-胺C28H31N5O453.578645944595
656247-17-5NintedanibBIBF 1120C31H33N5O4539.62482714653
728033-96-3Osi-930OSI930 抑制剂C22H16F3N3O2S443.441554069519
183320-51-6Desmethyl Erlotinib hydrochloride2-[[4-[(3-乙炔基苯基)氨基]-7-(2-甲氧基乙氧基)-6-喹唑啉基]氧]乙醇盐酸盐C21H22ClN3O4415.870084285736
196868-63-0PQ401PQ401 抑制剂C18H16ClN3O2341.791543006897
1061353-68-1PND-11862-(2-(2-甲氧基-4-吗啉代苯基氨基)-5-(三氟甲基)吡啶-4-基氨基)-N-甲基苯甲酰胺C25H26F3N5O3501.500855922699
477575-56-7Pha-665752(2R)-1-[[5-[(Z)-[5-[[(2,6-二氯苯基)甲基]磺酰]-1,2-二氢-2-氧代-3H-吲哚-3-亚基]甲基]-2,4-二甲基-1H-吡咯-3-基]羰基]-2-(1-吡咯烷甲基)吡咯烷C32H34Cl2N4O4S641.607764720917
444731-52-6Pazopanib帕唑帕尼C21H23N7O2S437.518021821976
257933-82-7Pelitinib培利替尼C24H23ClFN5O2467.923127412796
956905-27-4PF-042179032-[4-[1-(喹啉-6-甲基)-1H-[1,2,3]三唑并[4,5-B]吡嗪-6-基]-1H-吡唑-1-基]乙醇C19H16N8O372.383341789246
1092788-83-4PP121PP 121 *C17H17N7319.363781690598
717906-29-1PF-431396N-甲基-N-[2-[[[2-[(2-氧代-2,3-二氢-1H-吲哚-5-基)氨基]-5-三氟甲基嘧啶-4-基]氨基]甲基]苯基]甲磺酰胺C22H21F3N6O3S506.500753164291
183322-45-4PD153035 HydrochloridePD153035 抑制剂C16H15BrClN3O2396.66620182991
194423-15-9PD168393N-[4-[(3-溴苯基)氨基]-6-喹唑啉基]-2-丙烯酰胺C17H13BrN4O369.215322256088
635702-64-6Pazopanib hydrochloride盐酸帕唑帕尼C21H24ClN7O2S473.978960990906