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Diastereoselective radical mediated alkylation of a chiral glycolic acid derivative†‡
Liliana Parra Rapado,Philippe Renaud
Organic & Biomolecular Chemistry Pub Date : 05/24/2011 00:00:00 , DOI:10.1039/C1OB05230F
Abstract

Radical alkylation of 2-(tert-butyl)-2-methyldioxolan-4-one, a chiral equivalent of glycolic acid, occurs with good to high diastereoselectivity that compares favorably with the corresponding enolate alkylation. The importance of the position of the transition state position, early or late, is highlighted.

Graphical abstract: Diastereoselective radical mediated alkylation of a chiral glycolic acid derivative
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