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First enantiospecific synthesis of marine sesquiterpene quinol akaol A†‡
Enrique Alvarez-Manzaneda,Rachid Chahboun,Esteban Alvarez,Antonio Fernández,Ramón Alvarez-Manzaneda,Ali Haidour,Jose Miguel Ramos,Ali Akhaouzan
Chemical Communications Pub Date : 11/09/2011 00:00:00 , DOI:10.1039/C1CC14608D
Abstract

The first enantiospecific synthesis of akaol A, a marine sesquiterpene quinol, has been achieved. Key steps of the synthetic sequence are the oxidative degradation of (−)-sclareol to a dinorlabdane ketoester, mediated by the ozone–lead(IV) acetate system, the diastereoselective α-methylation of a ketoaldehyde, followed by an intramolecular aldol condensation and the further Diels–Alder cycloaddition of a dienol ether.

Graphical abstract: First enantiospecific synthesis of marine sesquiterpene quinol akaol A
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