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A new phosphonate pendant-armed cross-bridged tetraaminechelator accelerates copper(ii) binding for radiopharmaceutical applications†
Dannon J. Stigers,Riccardo Ferdani,Gary R. Weisman,Edward H. Wong,Carolyn J. Anderson,James A. Golen,Curtis Moore,Arnold L. Rheingold
Dalton Transactions Pub Date : 12/15/2009 00:00:00 , DOI:10.1039/B920871B
Abstract

A phosphonate pendant-armed cross-bridged cyclam chelator has been synthesized, complexed to Cu(II), radiolabeled with 64Cu under mild conditions, and its biodistribution studied.

Graphical abstract: A new phosphonate pendant-armed cross-bridged tetraamine chelator accelerates copper(ii) binding for radiopharmaceutical applications
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