Highly effective copper-catalyzed decarboxylative coupling of aryl halides with alkynyl carboxylic acids†
Xiaoming Qu,Tingyi Li,Peng Sun,Yan Zhu,Hailong Yang,Jincheng Mao
Organic & Biomolecular Chemistry Pub Date : 08/25/2011 00:00:00 , DOI:10.1039/C1OB05969F
Abstract

We have developed a highly effective copper-catalyzed decarboxylative coupling of alkynylcarboxylic acids with various aryl and alkyl halides at 2 mol% loading of copper. This method is simple, economical and practical for the synthesis of disubstituted alkyne compounds.

Graphical abstract: Highly effective copper-catalyzed decarboxylative coupling of aryl halides with alkynyl carboxylic acids