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Regiospecific synthesis of 3,4-disubstituted thiophenes
Chemical Communications Pub Date : 01/01/1900 00:00:00 , DOI:10.1039/CC9960000339
Abstract

3,4-Bis(trimethylsilyl)thiophene and several other 3,4-disubstituted thiophenes are synthesised by an unprecedented intermolecular cycloaddition窶田ycloreversion procedure between disubstituted acetylenes and 4-methyl- or 4-phenyl-thiazole; 3,4-bis(trimethylsilyl)thiophene undergoes consecutive regiospecific mono-ipso-iodination and palladium-catalysed reactions to provide unsymmetrically 3,4-disubstituted thiophenes.

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