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Synthetic chemistry-led creation of a difluorinated biaryl ether non-nucleoside reverse transcriptase inhibitor†
Lyn H. Jones,Amy Randall,Oscar Barba,Matthew D. Selby
Organic & Biomolecular Chemistry Pub Date : 10/02/2007 00:00:00 , DOI:10.1039/B714091F
Abstract

In the process of developing a series of novel, fluorinated biaryl ether NNRTIs, we fortuitously discovered derivative 20, which possesses excellent potency against both wild-type and clinically relevant mutations of the reverse transcriptase enzyme.

Graphical abstract: Synthetic chemistry-led creation of a difluorinated biaryl ether non-nucleoside reverse transcriptase inhibitor
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