960化工网
Synthesis and molecular structure of new acyclic analogues of nucleotides with a 1,2-alkadienic skeleton
Valery K. Brel,Vitaly K. Belsky,Adam I. Stash,Valery E. Zavodnik,Peter J. Stang
Organic & Biomolecular Chemistry Pub Date : 10/27/2003 00:00:00 , DOI:10.1039/B309684J
Abstract

Reaction of 1-chloro-4-(diethoxyphosphonyl)alka-2,3-dienes 14,15 with purine and pyrimidine heterocyclic bases in the presence of cesium carbonate afforded new acyclic analogues of nucleotides containing a 1,2-alkadienic skeleton 18–23. Dealkylation of 18–23 furnished phosphonic acids 2a–f. In contrast, alkylation reaction with 1-chloro-4-(diethoxyphosphonyl)octa-2,3-diene 16 led to Z- and E- 1,3-alkadienic phosphonates 25a,b and 26a,b. A similar reaction with 1-chloro-4-(diethoxyphosphonyl)-2-methylbuta-2,3-diene 17 led to the elimination of hydrochloride and formation of 4-(diethylphosphonyl)-2-methylbut-1-en-3-yne 24. Molecular structures of new acyclic nucleotides 18 and 2f are determined by X-ray crystallographic analysis.

Graphical abstract: Synthesis and molecular structure of new acyclic analogues of nucleotides with a 1,2-alkadienic skeleton
平台客服
平台客服
平台在线客服