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Synthesis of novel molecular probes inspired by harringtonolide†
Vinayak Hegde,Marc Campitelli,Ronald J. Quinn,David Camp
Organic & Biomolecular Chemistry Pub Date : 05/03/2011 00:00:00 , DOI:10.1039/C1OB05299C
Abstract

A novel harringtonolide-inspired scaffold containing a cycloheptatriene ring and two fused cyclopentane rings has been synthesised from simple starting materials. The scaffold, containing a similar substitution pattern and relative stereochemistry to the complex diterpenoid, has been enumerated into a small library of derivatives. One of these library members has been converted into a sub-library of substituted triazoles using copper-catalysed azide-alkyne cycloaddition (click) chemistry. The scaffold may be useful in drug discovery or in the preparation of additional molecular probes for chemical biology.

Graphical abstract: Synthesis of novel molecular probes inspired by harringtonolide
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