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The dihydrofuran template approach to furofuran synthesis†
David J. Aldous,Andrei S. Batsanov,Dmitrii S. Yufit,Anne J. Dalençon,William M. Dutton,Patrick G. Steel
Organic & Biomolecular Chemistry Pub Date : 06/30/2006 00:00:00 , DOI:10.1039/B604952D
Abstract

Flash vacuum pyrrolysis of vinyl epoxides provides cis-dihydrofuran carboxylic esters in good yields and diastereoselectivities, which, on base-promoted epimerisation afford the complementary trans series. The compounds provide a viable template for a Lewis acid promoted cyclisation to provide the 2,6-diaryl-3,7-dioxabicyclo[3.3.0]octane core found in the furofuran series of natural lignans. This strategy is stereodivergent and can be controlled to provide the exo-exo, exo-endo or endo-endo stereochemistries. The approach has been exemplified in syntheses of the sesamyl furofurans (±)-epiasarinin and (±)-asarinin.

Graphical abstract: The dihydrofuran template approach to furofuran synthesis
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