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Accessing bridged bicyclic compounds or meta carbon-functionalized anilines from the dearomatization of anilines†
Linfei Wang,Shuo-En Wang,Weibin Wang,Renhua Fan
RSC Advances Pub Date : 02/26/2013 00:00:00 , DOI:10.1039/C3RA23224G
Abstract

The oxidative dearomatization of anilines was combined with a domino Michael addition, providing a series of nitrogen-containing bridged bicyclic compounds in moderate to excellent yields. The bridged bicyclic compound could be converted into the corresponding meta carbon-functionalized aniline derivative via a quinine-catalyzed tandem retro-oxa-Michael addition–aromatization reaction.

Graphical abstract: Accessing bridged bicyclic compounds or meta carbon-functionalized anilines from the dearomatization of anilines
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