An enantioselective double Diels–Alder approach to the tetracyclic framework of colombiasin A†
Jason H. Chaplin,Alison J. Edwards,Bernard L. Flynn
Organic & Biomolecular Chemistry Pub Date : 05/13/2003 00:00:00 , DOI:10.1039/B302522E
Abstract

The complex tetracyclic carbon skeleton of colombiasin A is conveniently accessed through an enantioselective intermolecular Diels–Alder–sulfoxide elimination–intramolecular Diels–Alder (DA–E–IMDA) sequence.

Graphical abstract: An enantioselective double Diels–Alder approach to the tetracyclic framework of colombiasin A