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Rational design of a cyclin A fluorescent peptide sensor†
Elena Pazos,Miguel Pérez,Hugo Gutiérrez-de-Terán,Mar Orzáez,Tatiana Guevara,José L. Mascareñas,M. Eugenio Vázquez
Organic & Biomolecular Chemistry Pub Date : 08/23/2011 00:00:00 , DOI:10.1039/C1OB06009K
Abstract

We report the design and development of a fluorescent sensor specifically designed to target cyclin A, a protein that plays a key role in the regulation of the cell cycle. Computational studies provide a molecular picture that explains the observed emission increase, suggesting that the 4-DMAP fluorophore in the peptide is protected from the bulk solvent when inserted into the hydrophobic binding groove of cyclin A.

Graphical abstract: Rational design of a cyclin A fluorescent peptide sensor
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