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Trifluoromethyl syn- or anti-γ-amino alcohols by one-pot solvent-free Mannich-type reactions under temperature control†
Stefania Fioravanti,Luca Parise,Alessia Pelagalli,Lucio Pellacani,Laura Trulli
RSC Advances Pub Date : 03/17/2015 00:00:00 , DOI:10.1039/C5RA01791B
Abstract

Starting from trifluoroacetaldehyde ethyl hemiacetal, chiral amines and suitable aldehydes, diastereomerically pure fluorinated syn- or anti-γ-amino alcohols can be obtained by a friendly one-pot solvent-free L-proline catalysed Mannich-type reaction only by changing the temperature.

Graphical abstract: Trifluoromethyl syn- or anti-γ-amino alcohols by one-pot solvent-free Mannich-type reactions under temperature control
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