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An organocatalytic approach to enantiomerically enriched α-arylcyclohexenones and cyclohexanones†‡
Sara Duce,María Jorge,Inés Alonso,José Luis García Ruano,M. Belén Cid
Organic & Biomolecular Chemistry Pub Date : 11/01/2011 00:00:00 , DOI:10.1039/C1OB06356A
Abstract

The presence of a p-nitrophenyl group converts acetone into an excellent and versatile nucleophile in organocatalytic processes, able to react with α,β-unsaturated aldehydes affording β-substituted α-arylcyclohexenones via a Michael reaction/aldol reaction/dehydration sequence, which occurs in good yields, ee up to 96% and complete diastereoselectivity. The resulting compounds are excellent synthons for the diastereoselective preparation of a variety of synthetically useful polysubstituted cyclohexanones and derivatives.

Graphical abstract: An organocatalytic approach to enantiomerically enriched α-arylcyclohexenones and cyclohexanones
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