An environmentally benign approach for the synthesis of 3,3′-pyrrolidonyl spirooxindole derivatives via a cascade Knoevenagel–Michael–cyclization multicomponent reaction†
Chengbin Yu,Hairong Lyu,Yan Cai,Xinyu Miao,Zhiwei Miao
RSC Advances Pub Date : 08/12/2013 00:00:00 , DOI:10.1039/C3RA44119A
Abstract

A series of 3,3′-pyrrolidonyl spirooxindole derivatives have been synthesized in good yields from the cascade Knoevenagel–Michael–cyclization multicomponent reaction of isatin, malononitrile and α-isothiocyanato imide in the presence of a catalytic amount of triethylamine “on water” assisted with ultrasonic irradiation. The advantages of this method include high efficiency, mild reaction conditions and environmentally benign reagents. The current process provides a simple and green method for creating diversity-oriented syntheses of this intriguing class of compounds with potential biological activities.

Graphical abstract: An environmentally benign approach for the synthesis of 3,3′-pyrrolidonyl spirooxindole derivatives via a cascade Knoevenagel–Michael–cyclization multicomponent reaction