960化工网
Asymmetric addition of α-branched cyclic ketones to allenamides catalyzed by a chiral phosphoric acid†
Xiaoyu Yang,F. Dean Toste
Chemical Science Pub Date : 01/19/2016 00:00:00 , DOI:10.1039/C5SC04202J
Abstract

We describe the asymmetric addition of unactivated α-branched cyclic ketones to allenamides catalyzed by a chiral phosphoric acid, generating an all-carbon quaternary stereocenter with broad substrate scope and high enantioselectivity. The products are easily transformed into their corresponding 1,5- and 1,4-ketoaldehyde derivatives, which are both important building blocks in organic synthesis.

Graphical abstract: Asymmetric addition of α-branched cyclic ketones to allenamides catalyzed by a chiral phosphoric acid
平台客服
平台客服
平台在线客服