Rhodium(ii)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines†
Hai Shang,Yu Tian,Jun Luo,Lingyu Li,Yefeng Tang,Zhongmei Zou
RSC Advances Pub Date : 03/17/2016 00:00:00 , DOI:10.1039/C6RA02923J
Abstract

A novel rhodium(II)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles has been developed, which enables the facile synthesis of various 4-functionalized tetrahydro-β-carbolines as well as relevant scaffolds from readily available starting materials.

Graphical abstract: Rhodium(ii)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines