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Artificial lantipeptides from in vitrotranslations†
Jack W. Szostak
Chemical Communications Pub Date : 04/28/2011 00:00:00 , DOI:10.1039/C0CC05663D
Abstract

We have devised a protocol for enzyme-free insertion of dehydroalanine, dehydrobutyrine and thioether crosslinks into translated peptides. In vitro translation using 4-selenalysine and 4-selenoisoleucine as substitutes for lysine and isoleucine yields peptides that can be converted to polycyclic structures using mild chemistry in water. This methodology presents a gateway for exploring the potential of artificial lantipeptides as scaffolds for drug development.

Graphical abstract: Artificial lantipeptides from in vitro translations
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