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Catalytic asymmetric synthesis of α- and β-amino phosphonic acid derivatives
Jun-An Ma
Chemical Society Reviews Pub Date : 02/10/2006 00:00:00 , DOI:10.1039/B517100H
Abstract

Catalytic asymmetric reactions provide one of the most powerful and economical synthetic approaches to a variety of enantiomerically enriched compounds. As being analogues of the corresponding α- and β-amino acids, optically active α- and β-amino phosphonic acid derivatives have found widespread use in medicinal chemistry and the pharmaceutical sciences. Using catalytic amounts of chiral materials, asymmetric synthesis of enantiomerically enriched α- and β-amino phosphonates has been a subject of growing interest. This tutorial review contains a compilation of the catalytic asymmetric synthetic methods developed to date and highlights their utility for obtaining these target compounds.

Graphical abstract: Catalytic asymmetric synthesis of α- and β-amino phosphonic acid derivatives
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