Carbocyclization of unsaturated thioesters under palladium catalysis†
Arun P. Thottumkara,Toshiki Kurokawa,J. Du Bois
Chemical Science Pub Date : 04/24/2013 00:00:00 , DOI:10.1039/C3SC50486G
Abstract

An intramolecular thioesterolefin cross-coupling reaction for the preparation of cyclic ketone structures from unsaturated thioesters is described. This method capitalizes on the unique reactivity of thioesters with low-valent palladium catalysts and copper(I) salts to form acyl-metal species. Trapping of such intermediates with alkene functional groups generates the corresponding exo-methylene cycloalkanone products. Unsaturated thioester substrates, which can be accessed using a suite of modern synthetic methods, can now be regarded as precursors to complex carbocyclic derivatives.

Graphical abstract: Carbocyclization of unsaturated thioesters under palladium catalysis