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Claisen rearrangements of equilibrating allylic azides†
Donald Craig,John W. Harvey,Alexander G. O'Brien,Andrew J. P. White
Organic & Biomolecular Chemistry Pub Date : 08/30/2011 00:00:00 , DOI:10.1039/C1OB05972F
Abstract

Equilibrating mixtures of allylic azide-containing allylic alcohols or allylic 2-tolylsulfonylacetic esters undergo Johnson–Claisen or Ireland–Claisen rearrangement reactions to give unsaturated γ-azidoesters and -acids, respectively. Decarboxylation of the acids under basic conditions gives azidosulfones, with moderate to high diastereoselectivity.

Graphical abstract: Claisen rearrangements of equilibrating allylic azides
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