2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. GABA Receptor
  4. GMQ

GMQ 是一种酸敏感离子通道调节剂，也是竞争性 GABAAR 拮抗剂。GMQ 优先、高效、竞争性地抑制 GABAA 受体。GMQ 可抑制 α1β2、α1β2γ2、α4β2γ2 和 α5β2γ2 型 GABAA 受体。GMQ 通过抑制 GABA 能神经传递增强神经兴奋性。GMQ 在肠道系统中具有抗组胺作用，可抑制胃酸分泌。

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GMQ

GMQ Chemical Structure

CAS No. : 716-11-0

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规格 是否有货
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GMQ 的其他形式现货产品:

Other Forms of GMQ:

GMQ 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GMQ is an acid-sensing ion channel modulator, competitive GABAAR antagonist. GMQ preferentially, potently, competitively inhibits GABAARs. GMQ inhibits α1β2, α1β2γ2, α4β2γ2 and α5β2γ2 GABAARs. GMQ enhances neuronal excitation through inhibition of GABAergic transmission. GMQ has anti-histamine effects in the enteric system, inhibiting gastric acid secretion[1].

分子量

201.23

Formula

C10H11N5
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GMQ 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GMQ716-11-02-Guanidine-4-methylquinazolineGABA ReceptorGamma-aminobutyric acid Receptorγ-Aminobutyric acid ReceptorHEK293Tmiceanti-histamineInhibitorinhibitorinhibit

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HY-139226
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