2. Others GPCR/G Protein Neuronal Signaling
  3. Reference Standards Cholecystokinin Receptor
  4. L-365260 (Standard)

L-365260 (Standard) 是 L-365260 (HY-106840) 的分析标准品。本产品用于研究及分析应用。L-365260 是一种口服有效的和选择性的非肽胃泌素和脑胆囊收缩素受体 (CCK-B) 拮抗剂，其 Kis 值分别为 1.9 nM 和 2.0 nM。L-365260 以立体选择性和竞争性方式与豚鼠胃胃泌素和脑 CCK 受体相互作用。L-365260 可增强 Morphine 缓解疼痛的活性，并防止 Morphine 耐受。

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L-365260 (Standard)

L-365260 (Standard) Chemical Structure

CAS No. : 118101-09-0

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L-365260 (Standard) 相关抗体

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CCKAR CCKBR

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

L-365260 (Standard) is the analytical standard of L-365260 (HY-106840). This product is intended for research and analytical applications. L-365260 is an orally active and selective antagonist of non-peptide gastrin and brain cholecystoKinin receptor (CCK-B), with Kis of 1.9 nM and 2.0 nM, respectively. L-365260 interacts in a stereoselective and competitive manner with guinea pig stomach gastrin and brain CCK receptors. L-365260 can enhance Morphine analgesia and prevents Morphine tolerance[1][2][3].

IC50 & Target

Ki: 1.9 nM (gastrin); 2.0 nM (CCK-B)[1].
分子量

398.46

Formula

C24H22N4O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

L-365260 (Standard) 相关分类

  • 摩尔计算器

  • 稀释计算器

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

L-365260 (Standard)118101-09-0Reference StandardsCholecystokinin ReceptorCCK ReceptorgastrinbraincholecystokininCCK-BanalgesiaInhibitorinhibitorinhibit

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