2. Metabolic Enzyme/Protease
  3. Phosphodiesterase (PDE)
  4. PAT-078

PAT-078 是一种 II 型自分泌运动因子 (ATX) 抑制剂。PAT-078 主要占据 ATX 的疏水口袋，堵塞疏水通道与催化位点之间的瓶颈区域，且不与催化位点的锌离子发生相互作用。

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PAT-078

PAT-078 Chemical Structure

CAS No. : 1682644-84-3

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PAT-078 相关抗体

Top Publications Citing Use of Products

查看 Phosphodiesterase (PDE) 亚型特异性产品:

查看所有亚型
PDE1 PDE2 PDE3 PDE4 PDE5 PDE6 PDE7 PDE9 PDE10 PDE11 PDE12 PDE8 Autotaxin

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PAT-078 is a type II autotaxin (ATX) inhibitor. PAT-078 mainly occupies the hydrophobic pocket of ATX, blocks the bottleneck region between the hydrophobic channel and the catalytic site, and does not interact with the zinc ion at the catalytic site[1].

体外研究
(In Vitro)

PAT-078 是一种 II 型人源 ATX 抑制剂，可占据该酶的疏水口袋并诱导口袋重构[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

PAT-078 相关抗体:
分子量

430.86

Formula

C25H16ClFN2O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

PAT-078 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PAT-0781682644-84-3PAT078PAT 078Phosphodiesterase (PDE)Autotaxinhydrophobic channelhydrophobic pocketcatalytic sitehuman ATX inhibitorATX/ENPP-2zinc ionsType II inhibitorInhibitorinhibitorinhibit

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产品名称：
PAT-078
目录号：
HY-126229
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