2. PROTAC Epigenetics
  3. PROTACs Histone Methyltransferase
  4. PROTAC EZH2 Degrader-22

PROTAC EZH2 Degrader-22 (compound 7) 是一款靶向 EZH2 的 PROTAC 蛋白降解剂。PROTAC EZH2 Degrader-22 可用于癌症相关研究。


(粉色: EZH2 配体 (HY-13470)；蓝色: Cereblon 配体 (HY-103596)；黑色: 连接子)。

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PROTAC EZH2 Degrader-22

PROTAC EZH2 Degrader-22 Chemical Structure

CAS No. : 2653338-66-8

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PROTAC EZH2 Degrader-22 相关抗体

Top Publications Citing Use of Products

查看 PROTACs 亚型特异性产品:

查看所有亚型
von Hippel-Lindau (VHL) Cereblon MDM2 cIAP1

查看 Histone Methyltransferase 亚型特异性产品:

查看所有亚型
EZH1 EZH2 DOT1L SMYD2 SMYD3 SUV39H2/KMT1B EHMT2/G9a/KMT1C EHMT1/GLP/KMT1D ASH1L/KMT2H SETDB1/KMT2G SETD2/KMT3A NSD2/MMSET/WHSC1 SETD7/KMT7 SETD8/KMT5A PRMT1 PRMT3 PRMT4 PRMT5 PRMT6 PRMT7 PRMT8

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PROTAC EZH2 Degrader-22 (compound 7) is a PROTAC protein degrader targeting EZH2. PROTAC EZH2 Degrader-22 is applicable to cancer-related research[1].

(Pink: EZH2 ligand (HY-13470); Blue: Cereblon ligand (HY-103596); Black: linker).

体外研究
(In Vitro)

PROTAC EZH2 Degrader-22 (化合物 7) 具有浓度和时间依赖性活性，与 CRBN 配体、蛋白酶体抑制剂或 NAE 抑制剂联合处理可逆转其降解作用；PRC2 亚基的 mRNA 水平未受影响，表明其不涉及转录调控[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

PROTAC EZH2 Degrader-22 相关抗体:
分子量

939.15

Formula

C54H66N8O7
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

PROTAC EZH2 Degrader-22 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PROTAC EZH2 Degrader-222653338-66-8PROTACsHistone Methyltransferaseproteasomal degradationubiquitinationEZH2PRC2 subunitsH3K27me2/3Cereblon (CRBN)EEDSUZ12RbAp48E3 ubiquitin ligaseInhibitorinhibitorinhibit

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产品名称：
PROTAC EZH2 Degrader-22
目录号：
HY-181323
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