产品货号:A808115
产品名称:AZD2014
Synonyms:3-[2,4-Bis[(3S)-3-methyl-4-morpholinyl]pyrido[2,3-d]pyrimidin-7-yl]-N-methylbenzamide; Vistusertib
CAS号:1009298-59-2
分子式:C₂₅H₃₀N₆O₃
Appearance:Light Yellow Solid
Melting Point:233-237ºC
分子量:462.54
Storage:-20°C
Solubility:Chloroform (Slightly), Methanol (Slightly)
Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
应用:AZD2014 is a dual mTORC1 and mTORC2 inhibitor. Studies show that AZD2014 induces growth inhibition and cell death in breast cancer cell lines, including ER+ cell lines.
参考文献:Guichard, S.M. et al.: Cancer Res., 71, 917 (2012);
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