产品编号:A540250
化学名称:Alk 5 Inhibitor II
别名:2-[3-(6-Methyl-2-pyridinyl)-1H-pyrazol-4-yl]-1,5-naphthyridine; E 616452; RepSox; SJN 2511
CAS号:446859-33-2
分子式:C₁₇H₁₃N₅
Appearance:Light Beige to Brown Solid
Melting Point:189 - 192°C
分子量:287.32
存储条件:4°C
溶解度:Chloroform (Slightly), Methanol (Slightly)
类别:Research Tools; Enzyme Activators and Inhibitors;
应用:Alk 5 Inhibitor II is a selective ATP competitive inhibitor of transforming growth factor-b (TGFb). A potential drug for the treatment of fibrosis and cancer.
参考文献:Ren, J. et al.: Eur. J. Med. Chem., 44, 4259 (2009)
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